SCHEMBL8561489

SCHEMBL8561489

Cc1cc(C)cc(C(=O)CNCC(CCO)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 2/20 0.35
MCHR1 Q99705 1/20 0.35
CYP26A1 O43174 1/20 0.34
S1PR2 O95136 2/20 0.34
S1PR4 O95977 2/20 0.34
S1PR3 Q99500 2/20 0.34
TACR1 P25103 1/20 0.34
POLB P06746 1/20 0.34
S1PR1 P21453 1/20 0.34
ITGAV P06756 1/20 0.34
TACR2 P21452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561494 1.00 HTT (0.37) HTTALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL8064776 0.90 ALDH1A1 (0.36) HTTALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL8064773 0.90 ALDH1A1 (0.36) HTTALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL8053257 0.86 ALDH1A1 (0.37) HTTALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL8063808 0.86 ALDH1A1 (0.37) HTTALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL6603767 0.82 LMNA (0.41) HTTALDH1A1LMNASMN1; SMN2
SCHEMBL13965263 0.82 LMNA (0.41) HTTALDH1A1LMNASMN1; SMN2
SCHEMBL8559422 0.78 UTS2R (0.37) LMNAPOLBITGAV
SCHEMBL8878961 0.78 UTS2R (0.37) LMNAPOLBITGAV
SCHEMBL6604797 0.77 SLC6A2 (0.40) HTTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025617-A1 SUBSTITUTED ARYL PIPERAZINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-06-18 WO disclosed
EP-0783498-A4 SUBSTITUTED ARYL PIPERAZINES AS NEUROKININ ANTAGONISTS MERCK & CO INC (US) 1998-04-15 EP disclosed
EP-0783498-A1 SUBSTITUTED ARYL PIPERAZINES AS NEUROKININ ANTAGONISTS MERCK & CO. INC. (US) 1997-07-16 EP disclosed
US-5607936-A USEFUL IN TREATMENT OF RESPIRATORY DISEASES MERCK & CO., INC. (US) 1997-03-04 US disclosed
WO-1996010568-A1 SUBSTITUTED ARYL PIPERAZINES AS NEUROKININ ANTAGONISTS MERCK & CO., INC. (US) 1996-04-11 WO disclosed