SCHEMBL6604386

SCHEMBL6604386

CCOc1cc(C2=NN(C(=O)c3cccc(NC(=O)c4cnccn4)c3)CCC2)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
NPC1 O15118 3/20 0.51
HPGD P15428 1/20 0.51
MAPT P10636 1/20 0.43
PKM P14618 3/20 0.43
LMNA P02545 3/20 0.43
ALDH1A1 P00352 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KMT2A Q03164 5/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 2/20 0.42
CFTR P13569 1/20 0.42
HTT P42858 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
TP53 P04637 1/20 0.41
PGR P06401 3/20 0.41
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602109 0.95 RAB9A (0.53) RAB9ASMN1; SMN2NPC1HPGDMAPT
SCHEMBL6602654 0.92 RAB9A (0.47) RAB9ASMN1; SMN2NPC1HPGDMAPT
SCHEMBL6602816 0.92 NPC1 (0.48) RAB9ASMN1; SMN2NPC1MAPTPKM
SCHEMBL146882 0.91 MAPK1 (0.46) RAB9ASMN1; SMN2NPC1MAPTPKM
SCHEMBL6603283 0.90 ALDH1A1 (0.43) RAB9ASMN1; SMN2NPC1HPGDMAPT
Hydrochloric Acid SCHEMBL7652761 0.90 MAPK1 (0.45) RAB9ASMN1; SMN2NPC1MAPTPKM
SCHEMBL6600753 0.89 SMN1; SMN2 (0.44) RAB9ASMN1; SMN2NPC1PKMLMNA
SCHEMBL6601657 0.89 RAB9A (0.47) RAB9ASMN1; SMN2NPC1HPGDPKM
SCHEMBL6601223 0.88 ALDH1A1 (0.44) RAB9ASMN1; SMN2NPC1MAPTPKM
SCHEMBL6582371 0.88 NPC1 (0.49) RAB9ASMN1; SMN2NPC1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922036-B1 ARYLALKANOYL PYRIDAZINES MERCK PATENT GMBH (DE) 2004-03-24 EP disclosed
EP-1143944-A3 USE OF ARYLALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-09-11 EP disclosed
EP-1143944-A2 USE OF ARYLALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
WO-2000059484-A2 USE OF ARYLALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2000-10-12 WO disclosed
EP-0922036-A1 ARYLALKANOYL PYRIDAZINES MERCK PATENT GmbH (DE) 1999-06-16 EP disclosed
WO-1998006704-A1 ARYLALKANOYL PYRIDAZINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed