SCHEMBL6604561

SCHEMBL6604561

CCOC(=O)c1nc2cc(-c3nc(C)c[nH]3)c([N+](=O)[O-])cc2nc1OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
MITF O75030 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 2/20 0.39
POLB P06746 2/20 0.39
HPGD P15428 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
GALR2 O43603 1/20 0.39
HSP90AA1 P07900 1/20 0.39
XBP1 P17861 1/20 0.39
CCR6 P51684 1/20 0.39
MAPT P10636 4/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
CHEK1 O14757 1/20 0.36
DAPK3 O43293 1/20 0.36
PRKD3 O94806 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603534 0.91 ALDH1A1 (0.36) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6602204 0.90 ALDH1A1 (0.36) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6605470 0.84 ALDH1A1 (0.34) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6601960 0.83 KMT2A (0.41) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6602436 0.83 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2LMNAPOLBMAPT
SCHEMBL6603788 0.82 ALDH1A1 (0.38) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6603316 0.82 ALDH1A1 (0.45) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6376052 0.82 ALDH1A1 (0.45) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6603403 0.81 MAPT (0.32) ALDH1A1MITFSMN1; SMN2LMNAPOLB
SCHEMBL6602557 0.81 KMT2A (0.38) ALDH1A1MITFSMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020453-B1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERIVATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2004-05-19 EP disclosed
US-6348461-B1 CENTRAL NERVOUS SYSTEM ANTAGONIST WITH HETEROCYCLIC SUBSTITUENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1020453-A1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERI VATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed