SCHEMBL6602436

SCHEMBL6602436

CCOC(=O)c1ccc(NC(=O)OCc2c[nH]c(-c3cc4nc(C(=O)OCC)c(OCC)nc4cc3[N+](=O)[O-])n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NAMPT P43490 1/20 0.40
GRIA1 P42261 1/20 0.40
GRIA2 P42262 1/20 0.40
GRIA3 P42263 1/20 0.40
GRIA4 P48058 1/20 0.40
MAPT P10636 5/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MAPK1 P28482 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
KMT2A Q03164 4/20 0.38
RECQL P46063 1/20 0.38
BLM P54132 1/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603788 0.93 ALDH1A1 (0.38) ALDH1A1GAASMN1; SMN2GRIA1GRIA2
SCHEMBL6603385 0.90 KMT2A (0.40) ALDH1A1GAASMN1; SMN2GRIA1GRIA2
SCHEMBL6602557 0.90 KMT2A (0.38) ALDH1A1GAASMN1; SMN2GRIA1GRIA2
SCHEMBL6382753 0.88 NAMPT (0.43) SMN1; SMN2NAMPTMAPTNPC1RAB9A
SCHEMBL6601960 0.88 KMT2A (0.41) ALDH1A1GAASMN1; SMN2MAPTKMT2A
SCHEMBL6631139 0.87 ALDH1A1 (0.40) ALDH1A1GAASMN1; SMN2NAMPTGRIA1
SCHEMBL6605453 0.83 GRIA1 (0.58) GRIA1GRIA2GRIA3GRIA4
SCHEMBL6603403 0.83 MAPT (0.32) ALDH1A1GAASMN1; SMN2MAPTNPC1
SCHEMBL6603534 0.83 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL6604561 0.83 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020453-B1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERIVATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2004-05-19 EP disclosed
US-6348461-B1 CENTRAL NERVOUS SYSTEM ANTAGONIST WITH HETEROCYCLIC SUBSTITUENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1020453-A1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERI VATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed