SCHEMBL6604782

SCHEMBL6604782

O=[N+]([O-])c1ccc(S(=O)(=O)Nc2ccc(N3CCNCC3)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.70
ADRB1 P08588 1/20 0.69
SIRT6 Q8N6T7 1/20 0.69
CA2 P00918 3/20 0.57
CA1 P00915 2/20 0.57
CA9 Q16790 2/20 0.56
CA12 O43570 1/20 0.56
HDAC1 Q13547 1/20 0.53
ALDH1A1 P00352 5/20 0.52
MAPT P10636 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
KDM4E B2RXH2 2/20 0.52
RECQL P46063 1/20 0.52
CYP3A4 P08684 1/20 0.52
HPGD P15428 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
LMNA P02545 3/20 0.51
USP2 O75604 1/20 0.51
HTR1A P08908 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336262 0.83 SIRT6 (1.00) ADRB1SIRT6ALDH1A1MAPTKDM4E
SCHEMBL7526992 0.83 SIRT6 (1.00) ADRB1SIRT6ALDH1A1MAPTKDM4E
SCHEMBL18553766 0.82 HTR6 (1.00) HTR6ADRB1ALDH1A1MAPTMEN1
SCHEMBL18553746 0.82 HTR6 (0.89) HTR6ADRB1CA2CA1CA9
Hydrogen Sulfide SCHEMBL28002215 0.82 SIRT6 (0.96) ADRB1SIRT6ALDH1A1MAPTKDM4E
Hydrochloric Acid SCHEMBL1814630 0.82 SIRT6 (0.96) ADRB1SIRT6ALDH1A1MAPTKDM4E
SCHEMBL6152151 0.82 SIRT6 (0.96) ADRB1SIRT6ALDH1A1MAPTKDM4E
SCHEMBL1496058 0.82 SIRT6 (0.96) ADRB1SIRT6ALDH1A1MAPTKDM4E
SCHEMBL6151805 0.82 SIRT6 (0.96) ADRB1SIRT6ALDH1A1MAPTRECQL
Hydrochloric Acid SCHEMBL18553777 0.81 HTR6 (0.86) HTR6ADRB1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729455-B1 INDOLE-DERIVED AZYLPIPERAZINES AS LIGANDS FOR 5HT1-LIKE RECEPTORS 5HT1B AND 5HT1D PF MEDICAMENT (FR) 2004-09-08 EP disclosed
EP-0729455-A1 INDOLE-DERIVED AZYLPIPERAZINES AS LIGANDS FOR 5HT1-LIKE RECEPTORS 5HT1B AND 5HT1D PIERRE FABRE MEDICAMENT (FR) 1996-09-04 EP disclosed
WO-1995014004-A1 INDOLE-DERIVED AZYLPIPERAZINES AS LIGANDS FOR 5HT1-LIKE RECEPTORS 5HT1B AND 5HT1D PIERRE FABRE MEDICAMENT (FR) 1995-05-26 WO disclosed