SCHEMBL6605625

SCHEMBL6605625

O=C(CNC1CCN(S(=O)(=O)Cc2ccccc2)CC1)N1CC[C@H](F)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.51
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
RAB9A P51151 1/20 0.48
LMNA P02545 2/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216016 0.80 DPP4 (0.62)
Hydrochloric Acid SCHEMBL5218957 0.80 DPP4 (0.61)
SCHEMBL6609010 0.73 EBP (0.54) ALDH1A1MAPTMAPK1
SCHEMBL8342174 0.72 HPGD (0.63) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL12208343 0.71 ALDH1A1 (0.68) ALDH1A1MAPTRAB9ALMNAHDAC3
Hydrochloric Acid SCHEMBL4438401 0.71 HPGD (0.61) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL27857138 0.70 NPSR1 (0.72) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL7239112 0.70 HPGD (0.65) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL28949192 0.70 HPGD (0.68) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL6606715 0.70 ALDH1A1 (0.48) ALDH1A1MAPTRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399433-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-03-24 EP claimed
WO-2003002553-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-01-09 WO claimed
EP-1399433-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-03-24 EP disclosed
WO-2003002553-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-01-09 WO disclosed