SCHEMBL6605965

SCHEMBL6605965

CC(C)CCN(C(=O)OC(C)(C)C)C(=O)N(C1CCCNCC1O)S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
STS P08842 1/20 0.36
KCNH2 Q12809 1/20 0.34
HTR6 P50406 4/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HSD11B1 P28845 2/20 0.33
RORC P51449 2/20 0.33
HSD11B2 P80365 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
MBTPS1 Q14703 1/20 0.33
NOS1 P29475 3/20 0.33
NOS2 P35228 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6605969 1.00 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3STSKCNH2
SCHEMBL6607474 0.85 KCNA5 (0.39) STSPSEN1PSEN2APH1BNCSTN
SCHEMBL6605208 0.84 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3HTR6RORC
SCHEMBL6605205 0.84 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3HTR6RORC
SCHEMBL5971586 0.82 REN (0.32) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL3955650 0.81 CTSL (0.36) SLC6A2SLC6A4SLC6A3STSRORC
SCHEMBL3955653 0.81 CTSL (0.36) SLC6A2SLC6A4SLC6A3STSRORC
SCHEMBL3955656 0.79 STS (0.35) SLC6A2SLC6A4SLC6A3STSHTR6
SCHEMBL6589031 0.78
SCHEMBL6610801 0.71 MBTPS1 (0.34) SLC6A2SLC6A4SLC6A3MBTPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed