SCHEMBL6606500

SCHEMBL6606500

COc1cnc(CCl)cc1OCCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 4/20 0.44
PDE4A P27815 3/20 0.44
PDE4B Q07343 3/20 0.44
PDE4C Q08493 3/20 0.44
ADRB2 P07550 1/20 0.43
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
MTNR1B P49286 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
EBP Q15125 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606792 0.93 SIGMAR1 (0.47) SIGMAR1EBPTMEM97
SCHEMBL6610798 0.88 PDE4A (0.48) PDE4DPDE4APDE4BPDE4CADRB2
SCHEMBL6606686 0.83 PDE4B (0.42) PDE4DPDE4APDE4BPDE4CADRB2
SCHEMBL6606488 0.81 CYP11B1 (0.48) SIGMAR1EBPTMEM97
SCHEMBL6609628 0.80 PDE4B (0.41) PDE4DPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL10369608 0.78 PDGFRB (0.49) MTNR1B
SCHEMBL7596772 0.77 HTR2A (0.51) MTNR1B
SCHEMBL27278144 0.77 ALDH1A1 (0.41)
SCHEMBL6605638 0.76 SIGMAR1 (0.47) SIGMAR1EBPTMEM97
Hydrochloric Acid SCHEMBL9687781 0.76 ALDH1A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882714-B1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS PHARMACEUTICAL CO (JP) 2004-03-03 EP disclosed
US-5935977-A PHOSPHODIESTERASE IV INHIBITORS, TUMOR NECROSIS FACTOR-ALPHA PRODUCTION INHIBITORS; TREATING INFLAMMATORY AND AUTOIMMUNE DISEASES SS PHARMACEUTICAL CO., LTD. (JP) 1999-08-10 US disclosed
EP-0882714-A1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS Pharmaceutical Co., Ltd. (JP) 1998-12-09 EP disclosed