SCHEMBL6606675

SCHEMBL6606675

CCCCOC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)N(C)C(=O)OCC)cc3)C(=O)O2)CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.47
ITGA2B P08514 7/20 0.47
GRM2 Q14416 2/20 0.41
PRSS1 P07477 6/20 0.40
PRSS2 P07478 6/20 0.40
PRSS3 P35030 6/20 0.40
F10 P00742 6/20 0.39
SIGMAR1 Q99720 8/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601149 0.94 ITGB3 (0.53) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6603276 0.93 ITGB3 (0.56) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6604810 0.92 ITGB3 (0.52) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL7308588 0.90 ITGB3 (0.49) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6600714 0.89 ITGB3 (0.48) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6606261 0.89 ITGB3 (0.48) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6601512 0.89 ITGB3 (0.46) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6600939 0.88 ITGB3 (0.50) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL6602176 0.86 ITGB3 (0.59) ITGB3ITGA2BGRM2PRSS1PRSS2
SCHEMBL7310352 0.86 ITGB3 (0.47) ITGB3ITGA2BGRM2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed