SCHEMBL6606946

SCHEMBL6606946

CNNc1ncc(C(=O)O)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HCAR3 P49019 1/20 0.41
HCAR2 Q8TDS4 3/20 0.41
NAPRT Q6XQN6 1/20 0.41
TTR P02766 1/20 0.40
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
POLB P06746 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MGAM O43451 1/20 0.37
GRM5 P41594 2/20 0.36
LRRK2 Q5S007 1/20 0.36
TPMT P51580 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL476528 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EHCAR3HCAR2NAPRT
SCHEMBL31132753 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EHCAR3HCAR2NAPRT
SCHEMBL9648858 0.80 ALDH1A1 (0.43) ALDH1A1KDM4EHCAR3HCAR2NAPRT
SCHEMBL476556 0.77 MAPT (0.48) ALDH1A1KDM4EHCAR3GAAPOLB
SCHEMBL25933680 0.76 HCAR3 (0.54) ALDH1A1HCAR3POLB
SCHEMBL2421299 0.74 ALDH1A1 (0.41) ALDH1A1HCAR3HCAR2NAPRTTTR
SCHEMBL3635781 0.74 HCAR3 (0.54) HCAR3MGAMGRM5SMN1; SMN2MEN1
SCHEMBL3635976 0.74 GRM5 (0.51) KDM4EGAATDP1POLBHSD17B10
SCHEMBL990334 0.73 GRM5 (0.58) TDP1POLBGRM5SMN1; SMN2MEN1
SCHEMBL1105964 0.73 HCAR2 (0.47) ALDH1A1KDM4EHCAR3HCAR2NAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458684-A2 THERAPEUTIC HETEROCYCLES AstraZeneca AB (SE) 2004-09-22 EP disclosed
WO-2003051276-A2 THERAPEUTIC HETEROCYCLES ASTRAZENECA AB (SE) 2003-06-26 WO disclosed