SCHEMBL476556

SCHEMBL476556

O=C(O)c1cnc(NNC(=O)c2ccccc2)c(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
PTGS2 P35354 4/20 0.48
GAA P10253 5/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
HCAR3 P49019 1/20 0.46
MAPK1 P28482 2/20 0.44
PSMD14 O00487 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
ALDH1A1 P00352 3/20 0.43
TP53 P04637 1/20 0.42
MGAM O43451 1/20 0.42
TLR7 Q9NYK1 1/20 0.41
KCNQ3 O43525 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456000 0.82 MEN1 (0.44) MAPTSMN1; SMN2MEN1KMT2ANPSR1
SCHEMBL3635781 0.78 HCAR3 (0.54) SMN1; SMN2MEN1KMT2AHCAR3NPC1
SCHEMBL6606946 0.77 ALDH1A1 (0.41) MAPTSMN1; SMN2MEN1KMT2ANPSR1
SCHEMBL4756002 0.76 ALDH1A1 (0.39) MAPTSMN1; SMN2MEN1KMT2ANPSR1
SCHEMBL4704630 0.75 ALDH1A1 (0.38) MAPTSMN1; SMN2MEN1KMT2ANPSR1
SCHEMBL31132753 0.75 ALDH1A1 (0.47) MAPTMEN1KMT2AGAAKDM4E
SCHEMBL476528 0.75 ALDH1A1 (0.47) MAPTMEN1KMT2AGAAKDM4E
SCHEMBL21138873 0.73 PTGS2 (0.53) SMN1; SMN2MEN1KMT2APTGS2GAA
SCHEMBL6385971 0.72 ALDH1A1 (0.44) MAPTSMN1; SMN2GAAALDH1A1
SCHEMBL9648858 0.71 ALDH1A1 (0.43) SMN1; SMN2MEN1KMT2AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410857-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN Merck Sharp & Dohme Corp. (US) 2012-02-01 EP disclosed
WO-2010111058-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK SHARP & DOHME CORP. (US) 2010-09-30 WO disclosed