SCHEMBL6607136

SCHEMBL6607136

CCOC(=O)c1nc2cc(-n3ccc(=O)cc3)c([N+](=O)[O-])cc2nc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
MITF O75030 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
GRIA1 P42261 2/20 0.42
GRIA2 P42262 2/20 0.42
GRIA3 P42263 2/20 0.42
GRIA4 P48058 2/20 0.42
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
KCNMA1 Q12791 1/20 0.39
MAPT P10636 2/20 0.37
GRIK1 P39086 1/20 0.37
GRIK2 Q13002 1/20 0.37
GRIK3 Q13003 1/20 0.37
GRIK4 Q16099 1/20 0.37
GRIK5 Q16478 1/20 0.37
PTGER4 P35408 1/20 0.37
RAB9A P51151 1/20 0.37
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607856 0.85 MAPT (0.45) ALDH1A1MITFSMN1; SMN2GRIA1GRIA2
SCHEMBL6607045 0.81 ALDH1A1 (0.43) ALDH1A1MITFSMN1; SMN2PTGS1PTGS2
SCHEMBL6601059 0.81 GRIA1 (0.42) ALDH1A1MITFSMN1; SMN2GRIA1GRIA2
SCHEMBL6602490 0.80 GRIA1 (0.41) ALDH1A1MITFSMN1; SMN2GRIA1GRIA2
SCHEMBL6603200 0.79 GRIA1 (0.41) ALDH1A1MITFSMN1; SMN2GRIA1GRIA2
SCHEMBL6602596 0.79 ALDH1A1 (0.41) ALDH1A1MITFSMN1; SMN2PTGS1PTGS2
SCHEMBL6602905 0.79 GFER (0.52) ALDH1A1SMN1; SMN2MAPTLMNAHPGD
SCHEMBL8369082 0.77 PPARG (0.43) ALDH1A1MITFSMN1; SMN2PTGS1PTGS2
SCHEMBL6604726 0.76 ALDH1A1 (0.38) ALDH1A1MITFSMN1; SMN2PTGS1PTGS2
SCHEMBL5723168 0.74 GRIA1 (0.36) ALDH1A1GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020453-B1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERIVATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2004-05-19 EP disclosed
US-6348461-B1 CENTRAL NERVOUS SYSTEM ANTAGONIST WITH HETEROCYCLIC SUBSTITUENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1020453-A1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERI VATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed