SCHEMBL6608517

SCHEMBL6608517

N#Cc1cc(C(=O)CC(=O)Nc2cc(C(F)(F)F)c(N3CCC3)cc2NC(=O)O)ccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 2/20 0.40
POLB P06746 1/20 0.37
KDR P35968 2/20 0.36
SRPK2 P78362 1/20 0.36
SRPK1 Q96SB4 1/20 0.36
SRPK3 Q9UPE1 1/20 0.36
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.34
KDM4E B2RXH2 1/20 0.34
FASN P49327 1/20 0.34
THRB P10828 1/20 0.34
WDR5 P61964 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6612631 0.98 SCN10A (0.42) SCN10APOLBKDRSRPK2SRPK1
SCHEMBL7046359 0.92 KDM4E (0.44) MAPTSMN1; SMN2NPSR1LMNAKDM4E
SCHEMBL6163340 0.89 SCN10A (0.37) SCN10AKDRSRPK2SRPK1SRPK3
SCHEMBL6165622 0.88 SCN10A (0.39) SCN10AKDRSRPK2SRPK1SRPK3
SCHEMBL6685456 0.86 CHEK1 (0.38) SCN10APOLBMAPTSMN1; SMN2KDM4E
SCHEMBL6609589 0.86 MAPT (0.38) SCN10APOLBMAPTNPSR1
SCHEMBL6435938 0.82 KDR (0.34) SCN10APOLBKDRLMNATHRB
SCHEMBL6435489 0.82 THRB (0.41) MAPTSMN1; SMN2NPSR1LMNAKDM4E
SCHEMBL6610697 0.81 POLB (0.39) SCN10APOLBKDRSMN1; SMN2WDR5
SCHEMBL6607218 0.80 BDKRB1 (0.39) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed