SCHEMBL6610697

SCHEMBL6610697

CN(C)c1cc(NC(=O)O)c(NC(=O)CC(=O)c2ccnc(C#N)c2)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
KDR P35968 1/20 0.35
HDAC4 P56524 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
PARP14 Q460N5 1/20 0.32
SLC2A1 P11166 1/20 0.32
SLC2A3 P11169 1/20 0.32
SLC2A4 P14672 1/20 0.32
RAB9A P51151 2/20 0.32
WDR5 P61964 1/20 0.32
NPC1 O15118 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
IDH1 O75874 1/20 0.31
IDH2 P48735 1/20 0.31
SCN10A Q9Y5Y9 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607208 0.90 POLB (0.36) POLBKDRHDAC4HDAC6ALDH1A1
SCHEMBL6163566 0.89 KDR (0.35) POLBKDRHDAC4HDAC6
SCHEMBL6612157 0.86 ALDH1A1 (0.37) KDRALDH1A1MEN1KMT2APARP14
SCHEMBL6166120 0.81 AAK1 (0.36) POLBKDR
SCHEMBL6612631 0.81 SCN10A (0.42) POLBKDRSMN1; SMN2SCN10A
SCHEMBL6608517 0.81 SCN10A (0.40) POLBKDRWDR5SMN1; SMN2SCN10A
SCHEMBL27615910 0.81 POLB (0.43) POLB
SCHEMBL6607218 0.80 BDKRB1 (0.39) POLB
SCHEMBL7046359 0.79 KDM4E (0.44) ALDH1A1KMT2ASMN1; SMN2
SCHEMBL6435476 0.78 KDR (0.36) POLBKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed