SCHEMBL6608843

SCHEMBL6608843

CC(C)OC(=O)CON=C1C(=O)Nc2c1cc(-c1ccc(S(=O)(=O)N(C)C)cc1)c1c2CN(C)CC1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.37
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31
MEN1 O00255 2/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 2/20 0.31
MAPK1 P28482 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 2/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610824 0.90 HTR6 (0.36) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL6607933 0.90 HTR6 (0.38) HTR6GRIA1GRIA2GRIA3GRIA4
Hydrochloric Acid SCHEMBL6607627 0.89 HTR6 (0.37) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL6608854 0.89 HTR6 (0.37) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL6610333 0.88 MAPT (0.34) GRIA1GRIA2GRIA3GRIA4MEN1
SCHEMBL6607562 0.86 HTR6 (0.39) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL8133111 0.84 HTR6 (0.42) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL20694135 0.82 HTR6 (0.39) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL8133241 0.82 HTR6 (0.43) HTR6GRIA1GRIA2GRIA3GRIA4
SCHEMBL4401527 0.82 HTR6 (0.43) HTR6GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869958-B1 NOVEL INDOLE-2,3-DIONE-3-OXIME DERIVATIVES NEUROSEARCH AS (DK) 2004-12-29 EP claimed
EP-1066037-B1 USE OF INDOLE-2,3-DIONE-3-OXIME DERIVATIVES AS AMPA ANTAGONISTS NEUROSEARCH AS (DK) 2004-12-29 EP claimed