SCHEMBL6609300

SCHEMBL6609300

CC(=O)Oc1sccc1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 3/20 0.36
HSD17B10 Q99714 4/20 0.36
ALDH1A1 P00352 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
USP2 O75604 1/20 0.34
GLA P06280 1/20 0.34
CYP19A1 P11511 1/20 0.34
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
PTK2 Q05397 1/20 0.33
CUL4A Q13619 1/20 0.33
KDM4E B2RXH2 2/20 0.32
TSHR P16473 2/20 0.32
ELANE P08246 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4634541 0.86 KMT2A (0.36) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL4607918 0.81 KDM4E (0.36) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL27617435 0.79 ESR1 (0.41) LMNAHSD17B10ALDH1A1MEN1KMT2A
SCHEMBL27997449 0.78 LMNA (0.38) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL10872973 0.78 KDM4E (0.41) RAB9ALMNAHSD17B10ALDH1A1MAPK1
SCHEMBL27673491 0.78 LMNA (0.42) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL11459102 0.76 KDM4E (0.38) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL27680682 0.76 KMT2A (0.41) RAB9ALMNAHSD17B10ALDH1A1MEN1
SCHEMBL27703251 0.76 POLB (0.39) RAB9ANPC1LMNAHSD17B10ALDH1A1
SCHEMBL27997381 0.74 TNFSF11 (0.43) RAB9ANPC1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104292242-B Pyrantel compound and preparation, as well as preparation method and application of pyrantel compound and preparation 广州必贝特医药技术有限公司 2017-05-17 CN claimed
CN-104292242-A Pyrantel compound and preparation, as well as preparation method and application of pyrantel compound and preparation GUANGZHOU BEBETTER MEDICINE TECHNOLOGY CO LTD 2015-01-21 CN claimed
CN-110114647-A Temperature detection material, temperature detection ink using same, temperature indicator, method for manufacturing temperature detection material, and article management system 株式会社日立产机系统 2019-08-09 CN disclosed
CN-107074873-A 7- (morpholinyl) -2- (N-piperazinyl) methylthioeno [2, 3-c ] pyridine derivatives as anticancer agents 纳科法尔马有限公司 2017-08-18 CN disclosed
CN-106918995-A Photosensitive polymer combination, photosensitive-resin layered product, resin pattern and cured film method of manufacturing pattern and display device 旭化成株式会社 2017-07-04 CN disclosed
CN-104292242-B Pyrantel compound and preparation, as well as preparation method and application of pyrantel compound and preparation 广州必贝特医药技术有限公司 2017-05-17 CN disclosed
CN-102971327-B There is the anti-inflammatory compound of multiple tyrosine-kinase enzyme inhibition activity and the pharmaceutical compositions containing these compounds KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2016-04-20 CN disclosed
CN-102232071-B Fused polycyclic compounds as protein kinase inhibitors NATIONAL HEALTH RESEARCH INSTITUTES (CN) 2016-03-23 CN disclosed
CN-105218560-A The synthesis technique of 7-bromo-4-diuril phenol also [3,2-D] pyrimidine SHANGHAI TITAN TECHNOLOGY CO LTD 2016-01-06 CN disclosed
CN-102741256-B Protein kinase is had to the bicyclic heteroaryl derivative of inhibit activities HANMI PHARM. CO.,LTD. (KR) 2015-12-02 CN disclosed
CN-102365277-B JUN N-terminal kinase inhibitors ELAN PHARMACEUTICALS, INC. (US) 2015-11-25 CN disclosed
EP-1461333-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP disclosed
CN-1437587-A Benzoxazepinones and their use as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-08-20 CN disclosed
WO-2003044009-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO disclosed
CN-1418199-A Pyrimidine-4-one derivatives as LDL-PLA2 inhibitors SMITHKLINE BEECHAM PLC (GB) 2003-05-14 CN disclosed
CN-1360582-A Quinazoline derivs. ASTRAZENECA UK LTD (GB) 2002-07-24 CN disclosed
CN-1040213-C Diaryl 5,6-fusedheterocyclic acids as leukotriene antagonists MERCK FROSCT CANADA INC (CA) 1998-10-14 CN disclosed
CN-1027369-C Excitatory amino acid antagonists MERRELL DOW PHARMA (US) 1995-01-11 CN disclosed
CN-1081440-A 2-aryl-5,6-ring-fused pyrimidines and weeding are used ROHM & HAAS (US) 1994-02-02 CN disclosed
CN-1047292-A EAA antagonists MERRELL DOW PHARMA (US) 1990-11-28 CN disclosed