SCHEMBL6609746

SCHEMBL6609746

CC1Oc2ccc(CNCc3cccc(CNCc4cccc(Cl)c4)c3)cc2N=C1N

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 7/20 0.54
NOS1 P29475 7/20 0.54
NOS2 P35228 6/20 0.54
PARP1 P09874 1/20 0.41
CHRM2 P08172 1/20 0.40
HDAC1 Q13547 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
ROCK2 O75116 1/20 0.37
SMARCA2 P51531 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6306275 0.99 NOS3 (0.56) NOS3NOS1NOS2PARP1CHRM2
SCHEMBL7002475 0.99 NOS3 (0.55) NOS3NOS1NOS2PARP1CHRM2
Hydrochloric Acid SCHEMBL7004141 0.98 NOS1 (0.57) NOS3NOS1NOS2PARP1CHRM2
Hydrochloric Acid SCHEMBL6302705 0.92 NOS1 (0.46) NOS3NOS1NOS2PARP1ROCK2
Hydrochloric Acid SCHEMBL6998683 0.91 NOS1 (0.61) NOS3NOS1NOS2CHRM2HDAC1
SCHEMBL6609190 0.90 NOS3 (0.43) NOS3NOS1NOS2PARP1CYP1A2
SCHEMBL6613613 0.90 NOS3 (0.45) NOS3NOS1NOS2PARP1CHRM2
SCHEMBL6610312 0.90 PARP1 (0.51) NOS3NOS1NOS2PARP1ROCK2
Hydrochloric Acid SCHEMBL6306096 0.89 NOS3 (0.45) NOS3NOS1NOS2PARP1CYP1A2
Hydrochloric Acid SCHEMBL6302923 0.89 NOS3 (0.46) NOS3NOS1NOS2PARP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114037-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AG (DE) 2004-05-12 EP claimed