SCHEMBL6610312

SCHEMBL6610312

CC1Oc2ccc(CNCc3cccc(CNCc4ccccc4)c3)cc2N=C1N

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.51
NOS3 P29474 5/20 0.42
NOS2 P35228 5/20 0.42
NOS1 P29475 5/20 0.42
ROCK1 Q13464 2/20 0.39
ROCK2 O75116 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
BCHE P06276 1/20 0.35
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6309880 0.99 PARP1 (0.50) PARP1NOS3NOS2NOS1ROCK1
SCHEMBL27466929 0.97 PARP1 (0.53) PARP1NOS3NOS2NOS1ROCK1
Hydrochloric Acid SCHEMBL7713375 0.96 PARP1 (0.52) PARP1NOS3NOS2NOS1ROCK1
Hydrochloric Acid SCHEMBL6302705 0.95 NOS1 (0.46) PARP1NOS3NOS2NOS1ROCK1
SCHEMBL6611984 0.92 PARP1 (0.45) PARP1NOS3NOS2NOS1ROCK1
SCHEMBL6608031 0.92 PARP1 (0.42) PARP1NOS3NOS2NOS1ROCK1
Hydrochloric Acid SCHEMBL6302797 0.91 PARP1 (0.44) PARP1NOS3NOS2NOS1ROCK1
Hydrochloric Acid SCHEMBL6302716 0.91 NOS1 (0.43) PARP1NOS3NOS2NOS1ROCK1
SCHEMBL6610687 0.90 PARP1 (0.42) PARP1NOS3NOS2NOS1ROCK1
SCHEMBL6609746 0.90 NOS3 (0.54) PARP1NOS3NOS2NOS1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114037-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AG (DE) 2004-05-12 EP claimed
EP-1114037-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES Schering Aktiengesellschaft (DE) 2001-07-11 EP claimed
WO-2000017173-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-30 WO claimed