SCHEMBL6610003

SCHEMBL6610003

Clc1ccccc1C1c2[nH]c3ccccc3c2CCN1/C=C/Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
STAT3 P40763 1/20 0.48
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
PPARG P37231 1/20 0.46
RAB9A P51151 1/20 0.46
LMNA P02545 4/20 0.45
ESR1 P03372 2/20 0.43
PGR P06401 1/20 0.43
GRIN2B Q13224 1/20 0.42
ABCG2 Q9UNQ0 3/20 0.42
ABCB1 P08183 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6609980 0.86 SIGMAR1 (0.53) ADRA1DADRA1AADRA1BLMNAESR1
SCHEMBL6609979 0.86 SIGMAR1 (0.53) ADRA1DADRA1AADRA1BLMNAESR1
SCHEMBL7154434 0.86 LMNA (0.59) ADRA1DADRA1AADRA1BLMNAESR1
SCHEMBL7154439 0.86 LMNA (0.59) ADRA1DADRA1AADRA1BLMNAESR1
SCHEMBL6951397 0.77 ABCG2 (0.48) KDM4EALDH1A1ADRA1DADRA1AADRA1B
SCHEMBL7492514 0.77 PDE5A (0.55)
SCHEMBL6599818 0.76 ABCB1 (0.46) ADRA1DADRA1AADRA1BLMNAABCG2
SCHEMBL6615462 0.73 PDE5A (0.54)
SCHEMBL7497181 0.72 ABCG2 (0.62) ALDH1A1LMNAABCG2ABCB1MAPT
SCHEMBL23875966 0.71 KIF11 (0.63) GAAKDM4ELMNAESR1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458679-A2 PYRROLIDINE DERIVATIVES AS PROSTAGLANDIN MODULATORS Applied Research Systems ARS Holding N.V. (AN) 2004-09-22 EP disclosed
WO-2003053923-A2 PYRROLIDINE DERIVATIVES AS PROSTAGLANDIN MODULATORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2003-07-03 WO disclosed