SCHEMBL6612948

SCHEMBL6612948

COc1cnc(CC#N)cc1OCCc1scnc1C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.45
CYP4F2 P78329 3/20 0.38
CYP4A11 Q02928 3/20 0.38
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HPGD P15428 4/20 0.37
MAPT P10636 1/20 0.33
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611559 0.85 ALDH1A1 (0.42) CHEK1CYP4F2CYP4A11ALDH1A1KMT2A
SCHEMBL6606145 0.84 ALDH1A1 (0.48) CHEK1CYP4F2CYP4A11ALDH1A1KMT2A
SCHEMBL6606573 0.77 PDE3B (0.36)
SCHEMBL6605638 0.77 SIGMAR1 (0.47)
SCHEMBL6608302 0.74 KDM4E (0.36) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL6584988 0.73 CHEK1 (0.41) CHEK1CYP4F2CYP4A11ALDH1A1HPGD
SCHEMBL6606686 0.73 PDE4B (0.42)
SCHEMBL6611068 0.71 HPGD (0.40) CHEK1CYP4F2CYP4A11ALDH1A1KMT2A
SCHEMBL6611074 0.71 HPGD (0.40) CHEK1CYP4F2CYP4A11ALDH1A1KMT2A
SCHEMBL4851694 0.70 HPGD (0.43) CHEK1CYP4F2CYP4A11ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882714-B1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS PHARMACEUTICAL CO (JP) 2004-03-03 EP disclosed
US-5935977-A PHOSPHODIESTERASE IV INHIBITORS, TUMOR NECROSIS FACTOR-ALPHA PRODUCTION INHIBITORS; TREATING INFLAMMATORY AND AUTOIMMUNE DISEASES SS PHARMACEUTICAL CO., LTD. (JP) 1999-08-10 US disclosed
EP-0882714-A1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS Pharmaceutical Co., Ltd. (JP) 1998-12-09 EP disclosed