SCHEMBL6616461

SCHEMBL6616461

CC(CCCCBr)(C(=O)OCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
TDP1 Q9NUW8 2/20 0.46
KMT2A Q03164 2/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
AMPD3 Q01432 2/20 0.46
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MMP8 P22894 1/20 0.43
MAPK1 P28482 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
TSHR P16473 2/20 0.42
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
MAOB P27338 1/20 0.41
CYP3A4 P08684 1/20 0.40
MEN1 O00255 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6620085 0.85 TDP1 (0.49) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL28774981 0.79 MBOAT4 (0.48) ALDH1A1TDP1KMT2AAMPD3MMP8
SCHEMBL1706652 0.77 ALDH1A1 (0.60) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL23501489 0.76 ALDH1A1 (0.58) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL19105239 0.76 ALDH1A1 (0.58) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL522510 0.76 ALDH1A1 (0.62) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL991531 0.76 ALDH1A1 (0.62) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL2016291 0.75 ALDH1A1 (0.46) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL12632940 0.75 ALDH1A1 (0.46) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL12632939 0.75 ALDH1A1 (0.46) ALDH1A1TDP1KMT2ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683781-B1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE METABASIS THERAPEUTICS INC (US) 2004-04-21 EP disclosed
US-5731432-A Inhibitors of adenosine monophosphate deaminase GENSIA SICOR INC. (US) 1998-03-24 US disclosed
EP-0683781-A4 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE. GENSIA PHARMA (US) 1997-05-28 EP disclosed
EP-0683781-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA PHARMACEUTICALS, INC. (US) 1995-11-29 EP disclosed
WO-1994018200-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA, INC. (US) 1994-08-18 WO disclosed