SCHEMBL6617619

SCHEMBL6617619

COc1ccc(S(=O)(=O)C(N)(OCc2ccccc2)[C@H](O)[C@H](Cc2ccccc2)NC(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 7/20 0.45
MMP9 P14780 4/20 0.45
MMP13 P45452 4/20 0.45
MMP2 P08253 5/20 0.44
MMP3 P08254 4/20 0.44
PDE4A P27815 4/20 0.44
PDE4B Q07343 4/20 0.44
PDE4C Q08493 4/20 0.44
PDE4D Q08499 4/20 0.44
CA2 P00918 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KEAP1 Q14145 1/20 0.40
CTSD P07339 1/20 0.40
BACE1 P56817 1/20 0.40
FPR2 P25090 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6618902 0.90 KLK5 (0.46) MMP1MMP9MMP13MMP2MMP3
SCHEMBL7563179 0.84 HTT (0.43) MMP1MMP9MMP13MMP2CA2
SCHEMBL4863780 0.81 KLK5 (0.45) MMP1MMP9MMP13
SCHEMBL6617093 0.79 ATM (0.43) CTSD
SCHEMBL7562033 0.77 REN (0.46) MMP1MMP9MMP13
SCHEMBL5772204 0.75 MMP1 (0.38) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6617625 0.73 MMP2 (0.52) MMP1MMP9MMP13MMP2MMP3
SCHEMBL1601535 0.73 HTT (0.37) MMP1MMP9MMP13MMP2MMP3
SCHEMBL7587059 0.72 MLNR (0.45) CTSD
SCHEMBL1602562 0.72 HTT (0.37) MMP1MMP9MMP13MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086076-B1 SULFONAMIDE INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMA (US) 2004-12-22 EP disclosed