SCHEMBL6619946

SCHEMBL6619946

C[C@@H](C(=O)O)c1ccc(C2CNC(=O)N2C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.41
TP53 P04637 3/20 0.40
MDM2 Q00987 1/20 0.40
PTGS1 P23219 11/20 0.40
LMNA P02545 3/20 0.40
CYP2C9 P11712 2/20 0.40
AKR1C3 P42330 2/20 0.40
CXCR1 P25024 2/20 0.40
CXCR2 P25025 2/20 0.40
NFKB1 P19838 2/20 0.40
ALB P02768 1/20 0.40
ESR1 P03372 1/20 0.40
ALOX5 P09917 1/20 0.40
RARB P10826 1/20 0.40
ADRB3 P13945 1/20 0.40
HTR2A P28223 1/20 0.40
NR1I3 Q14994 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
CXCL8 P10145 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6615817 1.00 PTGS2 (0.41) PTGS2TP53MDM2PTGS1LMNA
SCHEMBL59197 0.70 PTGS2 (0.74) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL2436189 0.70 APP (0.56) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL11468007 0.67 APP (0.64) PTGS2PTGS1LMNACYP2C9AKR1C3
Hexaprofen SCHEMBL2111016 0.66 APP (0.67) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL185702 0.65 PTGS2 (0.61) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL1711069 0.65 PTGS2 (0.61) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL4767889 0.65 PTGS2 (0.61) PTGS2PTGS1LMNACYP2C9AKR1C3
SCHEMBL5727201 0.65 CCNA2 (0.53) PTGS2TP53PTGS1LMNACYP2C9
SCHEMBL7542404 0.65 PTGS1 (0.60) PTGS2PTGS1LMNACYP2C9AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406899-A2 PHENYLACETAMIDO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS Pharmacia Italia S.p.A. (IT) 2004-04-14 EP disclosed
WO-2003008365-A2 PHENYLACETAMIDO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA S.P.A. (IT) 2003-01-30 WO disclosed