SCHEMBL6622232

SCHEMBL6622232

CCNC(=O)N1C(=O)NC(C)=C(C#N)C1c1cccc(OC)c1.CCNC(=O)N1C(=O)NC(C)=C(C#N)C1c1ccccc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
MAPT P10636 3/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
ADRA1D P25100 5/20 0.38
ADRA1A P35348 5/20 0.38
ADRA1B P35368 5/20 0.38
USP2 O75604 1/20 0.38
THRB P10828 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313253 0.91 MAPK1 (0.48) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6312877 0.88 KDM4E (0.38) ALDH1A1KDM4EGAAHPGDMAPT
SCHEMBL6314801 0.82 MAPT (0.46) MAPK1ALDH1A1KDM4EMAPTADRA1D
SCHEMBL6320798 0.81 ALDH1A1 (0.51) MAPK1ALDH1A1KDM4EGAAMAPT
SCHEMBL6312051 0.79 ALDH1A1 (0.41) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6321577 0.79 ADRA1D (0.43) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6312755 0.79 ALDH1A1 (0.51) MAPK1ALDH1A1KDM4EGAAHPGD
SCHEMBL6320378 0.78 KDM4E (0.42) ALDH1A1KDM4EGAAHPGDMAPT
SCHEMBL6321556 0.78 CACNA1C (0.41) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL6314301 0.77 ABCC9 (0.45) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373221-A4 NOVEL CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL MYERS SQUIBB CO (US) 2004-09-29 EP claimed
EP-1373221-A2 NOVEL CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES Bristol-Myers Squibb Company (US) 2004-01-02 EP claimed
WO-2002079149-A2 NOVEL CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-10-10 WO claimed