SCHEMBL6624876

SCHEMBL6624876

C#Cc1ccc([C]=O)c(-c2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.41
GABRA5 P31644 6/20 0.41
GABRA2 P47869 6/20 0.41
GABRB2 P47870 4/20 0.41
GABRA3 P34903 4/20 0.41
GABRG2 P18507 3/20 0.41
GABRB3 P28472 3/20 0.41
KDM4E B2RXH2 1/20 0.34
GALR3 O60755 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
BACE1 P56817 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CYP2A6 P11509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12760764 0.81 FFAR1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL3800243 0.79 GABRA1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL7608202 0.76 GABRA1 (0.40) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL10659983 0.76 GABRA1 (0.38) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL27933506 0.75 PTGDR2 (0.47) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL7608526 0.75 NPC1 (0.38) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL224641 0.74 CASP3 (0.42) ALDH1A1HPGDBACE1CYP2A6FFAR1
SCHEMBL6625935 0.74 PTGDR2 (0.45) ALDH1A1HPGDPTGDR2BACE1
SCHEMBL6628582 0.74 PTGDR2 (0.45) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL11415648 0.74 BACE1 (0.56) GABRA1GABRA5GABRA2GABRB2GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986384-A4 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIV PITTSBURGH (US) 2004-09-15 EP disclosed
EP-0986384-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 2000-03-22 EP disclosed
WO-1998050029-A1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIVERSITY OF PITTSBURGH (US) 1998-11-12 WO disclosed