SCHEMBL10659983

SCHEMBL10659983

C#Cc1ccc(-c2ccccc2)c(C#C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.38
GABRA5 P31644 3/20 0.38
GABRA2 P47869 3/20 0.38
GABRB2 P47870 3/20 0.38
GABRA3 P34903 2/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
BACE1 P56817 1/20 0.37
ALOX5 P09917 1/20 0.36
CYP2A6 P11509 2/20 0.35
ABCG2 Q9UNQ0 1/20 0.33
FFAR1 O14842 1/20 0.33
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33
PBRM1 Q86U86 1/20 0.33
ESR2 Q92731 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GALR3 O60755 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3800243 0.83 GABRA1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL28739756 0.82 NPC1 (0.42) BACE1ALOX5CYP2A6ESR2KDM4E
SCHEMBL15901560 0.81 BACE1 (0.44) BACE1ALOX5CYP2A6SMARCA2SMARCA4
SCHEMBL7608202 0.80 GABRA1 (0.40) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL6138312 0.78 ESR2 (0.53) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL9303383 0.78 PTGS1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL9420892 0.78 CYP2A6 (0.54) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL28757167 0.78 ALDH1A1 (0.48) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL1302811 0.76 CYP2A6 (0.48) GABRA5GABRA3GABRG2GABRB3BACE1
SCHEMBL7608526 0.76 NPC1 (0.38) GABRA1GABRA5GABRA2GABRB2GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101948365-A Preparation method of 1,4-diaryl-1,3-butadiyne UNIV TONGJI 2011-01-19 CN disclosed
US-4767797-A Photocurable compositions of poly(ethynylphenyl)acetylene, its copolymer and composition thereof ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1988-08-30 US disclosed