SCHEMBL6627796

SCHEMBL6627796

O=C(O)c1ccc(CCC2CNc3ccc(C#CCc4cccnc4)cc3C2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.37
HIF1A Q16665 3/20 0.35
EPAS1 Q99814 3/20 0.35
GAA P10253 1/20 0.35
FFAR1 O14842 2/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
FFAR4 Q5NUL3 1/20 0.33
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
TBXAS1 P24557 3/20 0.33
NLRP3 Q96P20 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257608 0.75 MMP13 (0.40) MMP13HIF1AEPAS1GAAFFAR1
SCHEMBL6231446 0.66 GAA (0.56) MMP13GAA
SCHEMBL8996251 0.66 TBXAS1 (0.58) GAATBXAS1
SCHEMBL6302654 0.66 MMP13 (0.82) MMP13SLC22A8
SCHEMBL6252956 0.64 MMP13 (0.49) MMP13HIF1AEPAS1GAASLC22A8
SCHEMBL6254871 0.64 MMP13 (0.40) MMP13SLC22A8
SCHEMBL5353235 0.64 TBXAS1 (0.62) GAATBXAS1
SCHEMBL11067952 0.61 TBXAS1 (0.67) GAATBXAS1
SCHEMBL6477654 0.61 MMP13 (0.52) MMP13SLC22A8
SCHEMBL6450511 0.60 MMP13 (0.48) MMP13FFAR1SLC22A8FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1434585-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2004-07-07 EP claimed
WO-2003032999-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2003-04-24 WO claimed