SCHEMBL6629960

SCHEMBL6629960

NC1(c2ccccc2)CCN(c2nc3cccc4c3n2CCC4=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.36
SCD O00767 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
AKT1 P31749 3/20 0.34
KCNH2 Q12809 1/20 0.33
GRM2 Q14416 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
PTPN11 Q06124 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6507301 0.99 PARP1 (0.35) PARP1SCDCNR1CNR2AKT1
SCHEMBL6504752 0.85 MLYCD (0.39) PARP1CNR1CNR2AKT1KCNH2
Hydrochloric Acid SCHEMBL6139500 0.83 PARP1 (0.55) PARP1
SCHEMBL7262771 0.80 AVPR1A (0.43) PARP1OPRM1OPRD1OPRK1
SCHEMBL6630805 0.77 PARP1 (0.43) PARP1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL6510200 0.76 PARP1 (0.42) PARP1KDM4EALDH1A1
SCHEMBL6630480 0.76 MAPT (0.40) PARP1KDM4EALDH1A1
SCHEMBL7257136 0.75 OPRM1 (0.37) PARP1KCNH2GRM2OPRM1OPRD1
Hydrochloric Acid SCHEMBL6505881 0.75 MAPT (0.39) PARP1KDM4EALDH1A1
SCHEMBL6508880 0.75 CCR4 (0.39) PARP1OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309594-B1 BENZIMIDAZOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2004-12-15 EP claimed
EP-1309594-B1 BENZIMIDAZOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2004-12-15 EP disclosed
CN-1446218-A Benzimidazole derivatives, their preparation and their therapeutic use SANOFI SYNTHELABO (FR) 2003-10-01 CN disclosed