Phosphoric Acid

Phosphoric Acid

SCHEMBL6630320

O=P(O)(O)O.c1cc(-c2nc3c4c(ncc3[nH]2)CCOC4)no1

nearest known ligand 0.88

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Phosphoric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
WNT3A P56704 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphoric Acid SCHEMBL29660482 0.99 WNT3A (0.34) WNT3ATNKS2
Phosphoric Acid SCHEMBL5880378 0.99 WNT3A (0.34) WNT3ATNKS2
SCHEMBL5880375 0.94 WNT3A (0.34) WNT3ATNKS2
Hydrochloric Acid SCHEMBL5880349 0.92 WNT3A (0.34) WNT3ATNKS2
SCHEMBL7299546 0.76 WNT3A (0.34) WNT3ATNKS2
Hydrochloric Acid SCHEMBL7304498 0.60
SCHEMBL7299920 0.59 TNKS (0.34) WNT3ATNKS2
SCHEMBL15663037 0.58 GUCY1B2 (0.34)
SCHEMBL7296866 0.58
SCHEMBL7304154 0.57 BACE1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723732-B1 2-(3-ISOXAZOLYL)-3,6,7,9-TETRAHYDROIMIDAZO(4,5-D)PYRANO(4,3-B) PYRIDINE, PHARMACEUTICALLY ACCEPTABLE SALT OR HYDRATE THEREOF AND AQUEOUS BASE INCLUDING 1-MENTHOL, ETHANOL, AND PHOSPHATE BUFFER WITH PH OF 3 TO 5 SHIONOGI & CO., LTD. (JP) 2004-04-20 US claimed
EP-1132094-A1 PERCUTANEOUSLY ADMINISTRABLE PREPARATIONS CONTAINING CEREBRAL FUNCTION ACTIVATORS SHIONOGI & CO., LTD. (JP) 2001-09-12 EP claimed
EP-1270578-A4 NOVEL PROCESS FOR PRODUCING FUSED IMIDAZOPYRIDINE DERIVATIVE AND NOVEL CRYSTAL FORM SHIONOGI & CO (JP) 2004-11-03 EP disclosed
US-6723732-B1 2-(3-ISOXAZOLYL)-3,6,7,9-TETRAHYDROIMIDAZO(4,5-D)PYRANO(4,3-B) PYRIDINE, PHARMACEUTICALLY ACCEPTABLE SALT OR HYDRATE THEREOF AND AQUEOUS BASE INCLUDING 1-MENTHOL, ETHANOL, AND PHOSPHATE BUFFER WITH PH OF 3 TO 5 SHIONOGI & CO., LTD. (JP) 2004-04-20 US disclosed
WO-2001074821-A1 NOVEL PROCESS FOR PRODUCING FUSED IMIDAZOPYRIDINE DERIVATIVE AND NOVEL CRYSTAL FORM SHIONOGI & CO., LTD. (JP) 2001-10-11 WO disclosed
EP-1132094-A1 PERCUTANEOUSLY ADMINISTRABLE PREPARATIONS CONTAINING CEREBRAL FUNCTION ACTIVATORS SHIONOGI & CO., LTD. (JP) 2001-09-12 EP disclosed