SCHEMBL6631019

SCHEMBL6631019

Nc1[c]ccc(N)c1-c1cccc(N)c1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.37
PTPRC P08575 1/20 0.37
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CD44 P16070 1/20 0.34
PDK2 Q15119 1/20 0.34
HSPA1A P0DMV8 1/20 0.33
PABPC1 P11940 1/20 0.33
MAOA P21397 2/20 0.32
FGR P09769 1/20 0.32
PIM1 P11309 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CSNK1D P48730 1/20 0.32
DYRK1A Q13627 1/20 0.32
HIPK2 Q9H2X6 1/20 0.32
CSNK1G1 Q9HCP0 1/20 0.32
MAOB P27338 1/20 0.32
DPP4 P27487 1/20 0.31
HSD17B10 Q99714 2/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934331 0.71
SCHEMBL560128 0.71 ALDH1A1 (0.56) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL28440948 0.70 ALDH1A1 (0.43) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL2931225 0.69 ALOX15 (0.46) ADORA2APTPRCALDH1A1L3MBTL1CD44
Hydrochloric Acid SCHEMBL4521251 0.69 ALDH1A1 (0.53) ADORA2APTPRCALDH1A1L3MBTL1CD44
Methane SCHEMBL22720568 0.69 ALDH1A1 (0.53) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL9478614 0.69 ALDH1A1 (0.48) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL28440398 0.67 CA1 (0.42) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL29905105 0.67 ALDH1A1 (0.42) ADORA2APTPRCALDH1A1L3MBTL1CD44
SCHEMBL28448451 0.67 ALDH1A1 (0.58) ADORA2APTPRCALDH1A1L3MBTL1CD44

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1417202-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2004-05-12 EP disclosed
WO-2002079186-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2002-10-10 WO disclosed