SCHEMBL6632372

SCHEMBL6632372

CC(C)N[C@@H](CS(=O)(=O)Cc1ccccc1)C(=O)NCCCC[C@H](O)c1nc2ccccc2o1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 8/20 0.37
PTPN2 P17706 5/20 0.37
ALDH1A1 P00352 1/20 0.37
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
PTGER4 P35408 2/20 0.35
TLR2 O60603 1/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
HPGD P15428 1/20 0.34
FAAH O00519 1/20 0.34
CES1 P23141 1/20 0.34
DAGLA Q9Y4D2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6632980 0.87 ALDH1A1 (0.41) PTPN1PTPN2ALDH1A1
SCHEMBL6062639 0.86 CASP1 (0.34) PTPN1PTPN2ALDH1A1MTNR1AMTNR1B
SCHEMBL6062634 0.86 CASP1 (0.34) PTPN1PTPN2ALDH1A1MTNR1AMTNR1B
SCHEMBL6063534 0.86 CTSS (0.38) PTPN1PTPN2ALDH1A1
SCHEMBL6632750 0.86 ALDH1A1 (0.39) PTPN1PTPN2ALDH1A1PTGER4
SCHEMBL6630204 0.86 ALDH1A1 (0.39) PTPN1PTPN2ALDH1A1PTGER4
SCHEMBL6632745 0.86 ALDH1A1 (0.39) PTPN1PTPN2ALDH1A1PTGER4
SCHEMBL6628449 0.85 MAPT (0.46) PTPN1ALDH1A1KMT2AHPGD
SCHEMBL6061712 0.85 MAPT (0.46) PTPN1ALDH1A1KMT2AHPGD
SCHEMBL6062952 0.85 DAGLA (0.52) ALDH1A1MTNR1AMTNR1BFAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed