SCHEMBL6632649

SCHEMBL6632649

NC(=O)c1ccccc1Sc1ncco1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.53
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
PARP1 P09874 1/20 0.37
CSNK1A1 P48729 1/20 0.37
TYRO3 Q06418 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
CDC7 O00311 1/20 0.36
CTSA P10619 1/20 0.36
NUDT1 P36639 1/20 0.36
TRPA1 O75762 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
METAP2 P50579 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29123449 0.81 MAPT (0.50) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL3077375 0.76 SIRT1 (0.77) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6647601 0.76 SIRT1 (0.53) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6630356 0.74 SIRT1 (0.50) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6633089 0.71 SIRT1 (0.48) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7706549 0.71 SIRT1 (0.48) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7695938 0.71 SIRT1 (0.74) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6632529 0.71 SIRT1 (0.47) SIRT1KDM4EPARP1MAPTCDC7
SCHEMBL10767952 0.70 GRM5 (0.52) KDM4EALDH1A1HPGDHSD17B10PARP1
SCHEMBL6630237 0.70 SIRT1 (0.53) SIRT1ALDH1A1HPGDHSD17B10PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480977-A2 SUBSTITUTED ARYL COMPOUNDS FOR TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-12-01 EP disclosed
WO-2003070728-A2 AZABICYCLO-SUBSTITUTED BENZOYLAMIDES AND THIOAMIDES FOR TREATMENT OF CNS-RELATED DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2003-08-28 WO disclosed