SCHEMBL7706549

SCHEMBL7706549

CC(=O)c1cnc(Sc2ccccc2C(N)=O)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.48
PARP1 P09874 4/20 0.36
FAAH O00519 2/20 0.36
NSD2 O96028 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
GLA P06280 1/20 0.34
ICAM1 P05362 1/20 0.34
SELE P16581 1/20 0.34
AKR1C1 Q04828 1/20 0.34
TRPA1 O75762 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630356 0.81 SIRT1 (0.50) SIRT1PARP1FAAHNSD2KDM4E
SCHEMBL6632529 0.80 SIRT1 (0.47) SIRT1PARP1KDM4EGLAMAPT
SCHEMBL6633089 0.78 SIRT1 (0.48) SIRT1PARP1FAAHKDM4EALDH1A1
SCHEMBL6632850 0.74 SIRT1 (0.65) SIRT1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3077375 0.72 SIRT1 (0.77) SIRT1PARP1KDM4EALDH1A1HPGD
SCHEMBL6632649 0.71 SIRT1 (0.53) SIRT1PARP1KDM4EALDH1A1HPGD
SCHEMBL6647601 0.69 SIRT1 (0.53) SIRT1PARP1KDM4EALDH1A1HPGD
SCHEMBL6630704 0.68 SIRT1 (0.70) SIRT1NSD2KDM4EALDH1A1HPGD
SCHEMBL6630988 0.68 SIRT1 (0.64) SIRT1PARP1KDM4EALDH1A1HPGD
SCHEMBL6633917 0.66 SIRT1 (0.53) SIRT1PARP1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002016357-A2 QUINUCLIDINE-SUBSTITUTED ARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO disclosed