SCHEMBL6635529

SCHEMBL6635529

CCOC(=O)Cn1c(C(O)c2ccc(C#N)cc2)nc2ccc(NS(=O)(=O)c3ccccc3)cc21

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 4/20 0.45
SMARCA2 P51531 1/20 0.43
S1PR1 P21453 7/20 0.41
IMPDH2 P12268 1/20 0.40
PKM P14618 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
BRD4 O60885 2/20 0.39
BRD1 O95696 2/20 0.39
BRD9 Q9H8M2 2/20 0.39
BRPF3 Q9ULD4 2/20 0.39
BRD7 Q9NPI1 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
ATIC P31939 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635874 0.94 BRPF1 (0.47) BRPF1SMARCA2S1PR1PKMNPSR1
SCHEMBL8145525 0.84 F2 (0.52) BRPF1SMARCA2IMPDH2PKMBRD4
SCHEMBL6635525 0.83 AR (0.48) BRPF1SMARCA2PKMNPSR1MEN1
SCHEMBL6634425 0.81 HCRTR2 (0.39) S1PR1NPSR1MEN1ALDH1A1KMT2A
SCHEMBL6633352 0.81 LMNA (0.40) S1PR1NPSR1MEN1ALDH1A1KMT2A
SCHEMBL6639700 0.78 IRAK4 (0.44) NPSR1MEN1ALDH1A1KMT2A
SCHEMBL8029744 0.78 F2 (0.60) BRPF1SMARCA2PKMBRD4BRD1
SCHEMBL6635871 0.77 BRPF1 (0.48) BRPF1SMARCA2PKMNPSR1MEN1
SCHEMBL8027014 0.77 F2 (0.48) BRPF1SMARCA2PKMBRD4BRD1
SCHEMBL6639199 0.77 HCRTR2 (0.39) S1PR1NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed