SCHEMBL6635611

SCHEMBL6635611

Nc1c(C=O)ccc2c1C(=O)c1ccccc1C2=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.62
MAOB P27338 1/20 0.62
MAPK1 P28482 8/20 0.59
SMN1; SMN2 Q16637 7/20 0.59
ALDH1A1 P00352 6/20 0.59
MEN1 O00255 6/20 0.59
KMT2A Q03164 6/20 0.59
MAPT P10636 6/20 0.59
L3MBTL1 Q9Y468 4/20 0.59
POLB P06746 4/20 0.59
RAB9A P51151 4/20 0.59
TDP1 Q9NUW8 4/20 0.59
CYP3A4 P08684 3/20 0.59
NPC1 O15118 3/20 0.59
MCL1 Q07820 3/20 0.59
LMNA P02545 2/20 0.59
THRB P10828 2/20 0.59
TSHR P16473 2/20 0.59
CASP3 P42574 1/20 0.59
HBB P68871 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10785129 0.91 MAOA (0.47) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL15864613 0.79 MAPT (0.62) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL10815291 0.77 MEN1 (0.55) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL3247246 0.77 ADORA2A (0.53) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL487001 0.77 MAOA (1.00) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL30129869 0.77 MAOA (1.00) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL30173417 0.77 ADORA2A (0.53) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
Ammonia Solution, Strong SCHEMBL6046897 0.76 MAOA (0.96) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL8777879 0.74 MAOA (0.67) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1
SCHEMBL591041 0.74 ALDH1A1 (1.00) MAOAMAOBMAPK1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1447430-A1 New monoanthraquinone azamethine dyes CLARIANT INTERNATIONAL LTD. (CH) 2004-08-18 EP claimed
EP-1447429-A1 New bisanthraquinone azomethine dyes CLARIANT INTERNATIONAL LTD. (CH) 2004-08-18 EP claimed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-1447430-A1 New monoanthraquinone azamethine dyes CLARIANT INTERNATIONAL LTD. (CH) 2004-08-18 EP disclosed
EP-1447429-A1 New bisanthraquinone azomethine dyes CLARIANT INTERNATIONAL LTD. (CH) 2004-08-18 EP disclosed
US-5382465-A Durability MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-01-17 US disclosed
EP-0300770-B1 Polarizing film containing an anthraquinonic colorant MITSUI TOATSU CHEMICALS (JP) 1994-10-19 EP disclosed
US-5252769-A Anthraquinonic colorant and polarizing film containing the colorant MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1993-10-12 US disclosed
EP-0300770-A2 Polarizing film containing an anthraquinonic colorant MITSUI TOATSU CHEMICALS, Inc. (JP) 1989-01-25 EP disclosed