SCHEMBL6638679

SCHEMBL6638679

COC(=O)[C@H](Cc1ccc([N+](=O)[O-])cc1)NC(=O)c1c(C)cccc1C

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.55
ITGB1 P05556 2/20 0.47
ITGA4 P13612 2/20 0.47
ATM Q13315 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
CA2 P00918 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
RAB9A P51151 1/20 0.46
ITGA2 P17301 1/20 0.45
ITGB7 P26010 1/20 0.45
LNPEP Q9UIQ6 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.44
SSTR3 P32745 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582622 0.92 ITGB1 (0.56) L3MBTL1ITGB1ITGA4ALDH1A1MAPT
SCHEMBL7429256 0.92 ITGB1 (0.56) L3MBTL1ITGB1ITGA4ALDH1A1MAPT
SCHEMBL6580118 0.92 ITGB1 (0.52) L3MBTL1ITGB1ITGA4ATMALDH1A1
SCHEMBL12889768 0.87 ITGB1 (0.49) ITGB1ITGA4ALDH1A1MAPTSMN1; SMN2
SCHEMBL3316636 0.87 ITGB1 (0.49) ITGB1ITGA4ALDH1A1MAPTSMN1; SMN2
SCHEMBL11907045 0.84 CA2 (0.62) ALDH1A1MAPTCA2SMN1; SMN2NPC1
SCHEMBL6585927 0.84 ITGB1 (0.45) L3MBTL1ITGB1ITGA4ALDH1A1MAPT
SCHEMBL6580706 0.84 MEN1 (0.42) L3MBTL1ITGB1ITGA4ATMALDH1A1
SCHEMBL6639159 0.83 L3MBTL1 (0.60) L3MBTL1ITGB1ITGA4ATMALDH1A1
SCHEMBL15258099 0.82 CA2 (0.57) L3MBTL1ATMALDH1A1MAPTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005445-B1 N-ALKANOYLPHENYLALANINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-05-26 EP disclosed
EP-1403247-A1 N-Alkanoylphenylalanine derivatives F.HOFFMANN-LA ROCHE AG (CH) 2004-03-31 EP disclosed
US-6229011-B1 BINDING INHIBITORS BETWEEN VASCULAR ADHESION MOLECULE-1 AND ALPHA. BETA.INTEGRIN; USEFUL FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES SUCH AS MULTIPLE SCLEROSIS, ASTHMA, AND INFLAMMATORY BOWEL DISEASE HOFFMAN-LA ROCHE INC. 2001-05-08 US disclosed
EP-1005445-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-07 EP disclosed
WO-1999010312-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-04 WO disclosed