SCHEMBL7429256

SCHEMBL7429256

COC(=O)C(Cc1ccc([N+](=O)[O-])cc1)NC(=O)c1c(C)cccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.56
ITGA4 P13612 15/20 0.56
ITGB7 P26010 7/20 0.56
ITGA2 P17301 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.47
NOS2 P35228 2/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582622 1.00 ITGB1 (0.56) ITGB1ITGA4ITGB7ITGA2L3MBTL1
SCHEMBL12889768 0.94 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA2NOS2
SCHEMBL3316636 0.94 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA2NOS2
SCHEMBL6638679 0.92 L3MBTL1 (0.55) ITGB1ITGA4ITGB7ITGA2L3MBTL1
SCHEMBL6585927 0.90 ITGB1 (0.45) ITGB1ITGA4ITGB7ITGA2L3MBTL1
SCHEMBL6580118 0.88 ITGB1 (0.52) ITGB1ITGA4ITGB7L3MBTL1ALDH1A1
SCHEMBL27541119 0.87 NOS2 (0.43) ITGB1ITGA4ITGB7ITGA2NOS2
SCHEMBL27541117 0.87 NOS2 (0.43) ITGB1ITGA4ITGB7ITGA2NOS2
SCHEMBL7432342 0.86 L3MBTL1 (0.64) ITGB1ITGA4ITGB7ITGA2L3MBTL1
SCHEMBL6639882 0.85 ITGB1 (0.60) ITGB1ITGA4ITGB7ITGA2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100369888-C N-alkanoylphenylalanine derivatives HOFFMANN LA ROCHE (CH) 2008-02-20 CN disclosed
CN-1281430-A N-alkanoylphenylalanine derivatives HOFFMANN LA ROCHE (CH) 2001-01-24 CN disclosed
EP-1005445-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-07 EP disclosed
WO-1999010312-A1 N-ALKANOYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-04 WO disclosed