SCHEMBL6642201

SCHEMBL6642201

O=C(Nc1cnccn1)c1cccnc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.67
SMN1; SMN2 Q16637 3/20 0.64
LMNA P02545 1/20 0.63
HIF1A Q16665 1/20 0.63
TSHR P16473 2/20 0.62
HSD17B10 Q99714 2/20 0.62
ALOX15 P16050 1/20 0.62
CASP1 P29466 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
NPC1 O15118 1/20 0.61
TP53 P04637 1/20 0.61
MAPT P10636 1/20 0.61
NFKB1 P19838 1/20 0.61
RAB9A P51151 1/20 0.61
NFKB2 Q00653 1/20 0.61
RELA Q04206 1/20 0.61
ROCK2 O75116 1/20 0.61
ROCK1 Q13464 1/20 0.61
HDAC1 Q13547 2/20 0.59
HDAC6 Q9UBN7 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45148 0.88 KMT2A (0.73) KMT2ASMN1; SMN2TSHRHSD17B10ALOX15
SCHEMBL29238994 0.87 KMT2A (0.71) KMT2ASMN1; SMN2TSHRHSD17B10ALOX15
SCHEMBL30533391 0.87 KMT2A (0.71) KMT2ASMN1; SMN2TSHRHSD17B10ALOX15
SCHEMBL6646471 0.85 RAB9A (0.70) KMT2ASMN1; SMN2LMNAHIF1ATSHR
SCHEMBL31414959 0.85 RAB9A (0.70) KMT2ASMN1; SMN2LMNAHIF1ATSHR
SCHEMBL3409741 0.83 KMT2A (0.66) KMT2ASMN1; SMN2LMNATSHRHSD17B10
SCHEMBL23015752 0.80 RAB9A (0.67) KMT2ASMN1; SMN2LMNAHIF1AHSD17B10
SCHEMBL23446461 0.80 MAPK8 (0.62) KMT2ASMN1; SMN2LMNAHIF1ANPC1
SCHEMBL18398740 0.80 TSHR (0.66) KMT2ASMN1; SMN2TSHRHSD17B10ALOX15
SCHEMBL23410523 0.80 MAPK8 (0.62) SMN1; SMN2LMNAHIF1AHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453831-A1 1H-PYRROLO(3,2-B)PYRIDINE-3-CARBOXYLIC ACID AMIDES Neurogen Corporation (US) 2004-09-08 EP claimed
WO-2003044018-A1 1H-PYRROLO[3,2-B]PYRIDINE-3-CARBOXYLIC ACID AMIDES NEUROGEN CORPORATION (US) 2003-05-30 WO claimed
WO-2025092884-A1 METHOD FOR TREATING LEUKEMIA 深圳市塔吉瑞生物医药有限公司 2025-05-08 WO disclosed
CN-109651359-B Substituted nicotinamide compound, pharmaceutical composition and application thereof 深圳市塔吉瑞生物医药有限公司 2021-06-22 CN disclosed