SCHEMBL6644141

SCHEMBL6644141

Cc1ccc(C2CNCCN2)nc1C

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
PARP1 P09874 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5088449 0.77 CCR1 (0.39) TLR9TLR8TLR7PARP1NOS3
SCHEMBL9733257 0.72 CYP3A4 (0.41) PARP1NOS2
SCHEMBL171615 0.72 CHEK1 (0.47)
SCHEMBL10080114 0.70 HTR2C (0.46) TLR9TLR8TLR7
SCHEMBL7306428 0.70 MEN1 (0.40) TLR9TLR8TLR7PARP1
SCHEMBL6764229 0.70 BMPR1B (0.33) TLR9TLR8TLR7PARP1NOS3
SCHEMBL6965088 0.69 HTR2A (0.37)
SCHEMBL9786097 0.69 HTR2A (0.37)
SCHEMBL27848286 0.69 HTR2C (0.39) TLR9TLR8TLR7PARP1
SCHEMBL526057 0.69 PRKCZ (0.38) TLR9TLR8TLR7PARP1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373247-A2 SPIROISOQUINOLINE COMPOUNDS, METHODS FOR THEIR PREPARATION AND INTERMEDIATES THEREOF TANABE SEIYAKU CO., LTD. (JP) 2004-01-02 EP disclosed
WO-2002079189-A2 SPIROISOQUINOLINE COMPOUNDS, METHODS FOR THEIR PREPARATION AND INTERMEDIATES TANABE SEIYAKU CO., LTD. (JP) 2002-10-10 WO disclosed