SCHEMBL9733257

SCHEMBL9733257

c1ccc2nc(C3CNCCN3)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.41
ALDH1A1 P00352 4/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPK1 P28482 2/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.41
HIF1A Q16665 1/20 0.41
CYP1A2 P05177 5/20 0.41
KDM4E B2RXH2 4/20 0.41
PMP22 Q01453 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
USP2 O75604 1/20 0.41
HTR3B O95264 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR1A P08908 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526057 0.80 PRKCZ (0.38) MEN1KMT2ASMN1; SMN2CYP1A2HTR2C
SCHEMBL6233129 0.79 CYP1A2 (0.41) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL27608178 0.79 BACE1 (0.41) KMT2AHTR2CSLC6A4PARP1BACE1
SCHEMBL27627374 0.79 BACE1 (0.41) HTR2CHTTPARP1NCF1BACE1
SCHEMBL28752901 0.79 HRH3 (0.37) NPC1RAB9AKMT2AHIF1AKDM4E
SCHEMBL16429508 0.79 TAAR1 (0.49) CYP3A4ALDH1A1NPC1RAB9AMEN1
SCHEMBL28800404 0.78 KDM4E (0.39) ALDH1A1MEN1KMT2AMAPTCYP1A2
SCHEMBL9317927 0.78 BACE1 (0.43) PARP1BACE1
SCHEMBL8918069 0.77 CYP2D6 (0.52) CYP3A4ALDH1A1NPC1RAB9AMEN1
SCHEMBL6233506 0.75 BMPR1B (0.36) CYP3A4ALDH1A1MAPK1CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120641-A Incubating with sample, determining radioactivity DAIICHI PURE CHEMICALS CO., LTD. (JP) 1992-06-09 US disclosed
EP-0435192-A2 Method for measurement of serotonin uptake sites and radioligand therefor DAIICHI PURE CHEMICALS CO. LTD. (JP) 1991-07-03 EP disclosed