SCHEMBL6644233

SCHEMBL6644233

CC(=O)N1CCc2cc(NC(=O)c3ccc(C)nc3N3CCC(C)CC3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.55
TP53 P04637 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
PDE7A Q13946 2/20 0.49
LMNA P02545 2/20 0.48
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
SCN10A Q9Y5Y9 2/20 0.46
NOTUM Q6P988 3/20 0.44
THRB P10828 1/20 0.42
SYK P43405 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646611 0.93 SCN10A (0.46) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6649216 0.89 CASP3 (0.44) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6645438 0.88 SCN10A (0.42) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6642943 0.84 PDE7A (0.40) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6649404 0.83 PDE7A (0.41) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6649155 0.83 PDE7A (0.41) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6646845 0.83 EIF2AK3 (0.42) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6647715 0.83 PDE7A (0.40) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6645593 0.83 MAPT (0.48) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL6642104 0.83 SCN10A (0.44) MAPTTP53SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040133008-A1 Amide compounds FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-08 US disclosed
WO-2004039795-A2 AMIDE COMPOUNDS FOR THE TREATMENT OF HYPERLIPIDEMIA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-05-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040133008-A1 Amide compounds APOB, APOL1, LDLR MAPT 4101/4885TP53 4513/4885SMN1; SMN2 1836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.