SCHEMBL6644355

SCHEMBL6644355

ON=C1CCc2sccc21

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.78
HPGD P15428 3/20 0.40
HTT P42858 3/20 0.40
LMNA P02545 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NOS2 P35228 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PLK4 O00444 1/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
PIM1 P11309 1/20 0.38
PDGFRA P16234 1/20 0.38
PRKACA P17612 1/20 0.38
LTK P29376 1/20 0.38
GRK5 P34947 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5455999 0.88 USP2 (0.92) USP2HPGDHTTLMNANPSR1
SCHEMBL3578599 0.88 USP2 (0.92) USP2HPGDHTTLMNANPSR1
SCHEMBL3578601 0.88 USP2 (0.92) USP2HPGDHTTLMNANPSR1
SCHEMBL9039199 0.72 USP2 (0.53) USP2HPGDHTTLMNANPSR1
SCHEMBL9039193 0.72 USP2 (0.53) USP2HPGDHTTLMNANPSR1
SCHEMBL17225406 0.69 NOS2 (0.45) USP2LMNANOS2PLK4CHEK1
SCHEMBL7934124 0.68 USP2 (0.48) USP2HPGDHTTLMNANPSR1
SCHEMBL7293034 0.68 USP2 (0.48) USP2HPGDHTTLMNANPSR1
SCHEMBL15219995 0.67 CES1 (0.50) USP2HPGDLMNANOS2PLK4
SCHEMBL9865315 0.64 USP2 (0.44) USP2HPGDNOS2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401830-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2004-03-31 EP disclosed
US-20030114666-A1 Having quinazolindione core structure; non-antibiotic resistance WARNER-LAMBERT COMPANY 2003-06-19 US disclosed
WO-2002102793-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2002-12-27 WO disclosed
WO-2001015677-A2 USE OF 5-HT1B/1D AGONISTS TO TREAT OTIC PAIN ALCON LABORATORIES, INC. (US) 2001-03-08 WO disclosed
US-5252749-A Binding to serotonin receptors 5HT3, 5HT1D and 5HT1B; hypotensive agents; cardiovascular and psychological disorders ELF SANOFI (FR) 1993-10-12 US disclosed
US-5252749-A Binding to serotonin receptors 5HT3, 5HT1D and 5HT1B; hypotensive agents; cardiovascular and psychological disorders ELF SANOFI (FR) 1993-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114666-A1 Having quinazolindione core structure; non-antibiotic resistance ABCC1, RPS6KA1, SIGMAR1 USP2 4179/4885HPGD 633/4885HTT 4546/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.