SCHEMBL6645857

SCHEMBL6645857

CCCCCNc1c2c(nn1C)N(c1c(C)cc(C)cc1C)CCC2

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.36
CRHR1 P34998 2/20 0.35
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NR1I2 O75469 1/20 0.32
BCHE P06276 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5043421 0.92 CRHR1 (0.31) CRHR1POLB
SCHEMBL6645359 0.92 ACHE (0.35) ACHECRHR1HPGDNPSR1KDM4E
SCHEMBL5039764 0.84 CRHR1 (0.32) CRHR1
SCHEMBL5048460 0.84 CRHR1 (0.39) CRHR1HPGDNPSR1KDM4ELMNA
SCHEMBL5039172 0.82 GAA (0.44) CRHR1NPSR1POLBHTTSMN1; SMN2
SCHEMBL5045685 0.80 CRHR1 (0.39) CRHR1
SCHEMBL6053104 0.80 CRHR1 (0.47) ACHECRHR1HPGDKDM4ELMNA
SCHEMBL6303475 0.79 CRHR1 (0.47) ACHECRHR1KDM4ELMNAPOLB
SCHEMBL5522195 0.79 CRHR1 (0.33) CRHR1NR1I2
SCHEMBL5043583 0.78 TSHR (0.38) CRHR1HPGDKDM4EPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453832-A1 RING FUSED PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2004-09-08 EP claimed
WO-2003048160-A1 RING FUSED PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-06-12 WO claimed