SCHEMBL6647355

SCHEMBL6647355

NC(Cc1nc(O)c(O)c(C(=O)NCc2ccc(F)cc2)n1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
ERCC1 P07992 1/20 0.43
FEN1 P39748 1/20 0.43
ERCC4 Q92889 1/20 0.43
ALDH1A1 P00352 4/20 0.42
LMNA P02545 2/20 0.42
PTGER4 P35408 1/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.41
CXCR4 P61073 1/20 0.41
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6647885 0.85 SMN1; SMN2 (0.42) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL5259936 0.85 SMN1; SMN2 (0.47) ERCC1FEN1ERCC4ALDH1A1HPGD
Hydrochloric Acid SCHEMBL5255058 0.84 SMN1; SMN2 (0.46) ERCC1FEN1ERCC4ALDH1A1HPGD
SCHEMBL6647317 0.82 ALDH1A1 (0.44) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL5129033 0.82 ALDH1A1 (0.50) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL5127722 0.82 ALDH1A1 (0.46) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL6648519 0.82 KCNE1 (0.44) KMT2AERCC1FEN1ERCC4ALDH1A1
SCHEMBL5127980 0.81 CXCR4 (0.53) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL5117167 0.81 LMNA (0.49) KMT2ACYP1A2CYP2C19ERCC1FEN1
SCHEMBL5128003 0.81 ALDH1A1 (0.50) KMT2AERCC1FEN1ERCC4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2004-08-04 EP claimed
WO-2003035076-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO claimed
EP-1441734-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2004-08-04 EP disclosed
WO-2003035076-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO disclosed