SCHEMBL6649262

SCHEMBL6649262

NC(=O)c1nc(-c2ccc([N+](=O)[O-])s2)nc(O)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 1/20 0.41
HSP90AA1 P07900 1/20 0.41
RECQL P46063 1/20 0.41
CYP2A6 P11509 1/20 0.39
ATM Q13315 1/20 0.34
ALOX5 P09917 1/20 0.34
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
TSHR P16473 1/20 0.33
NR1D1 P20393 1/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA12 O43570 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5125073 0.77 L3MBTL1 (0.45) ALDH1A1MAPTLMNAKMT2AL3MBTL1
SCHEMBL6648977 0.72 CYP2A6 (0.43) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL6644722 0.71 ERCC1 (0.57) ALDH1A1MAPTKMT2AKDM4ERAB9A
SCHEMBL9777499 0.65 CYP2A6 (0.56) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL30142861 0.65 BCAT2 (0.45) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL2118284 0.65 ATM (0.55) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL6068076 0.64 CYP2A6 (0.49) ALDH1A1MAPTLMNAKMT2ACYP2A6
SCHEMBL6643744 0.64 IKBKB (0.51) KMT2AKDM4EMEN1GAAJAK2
SCHEMBL6649260 0.62 CYP2A6 (0.41) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL6649184 0.62 ADORA2A (0.41) RAB9AHSP90AA1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2004-08-04 EP disclosed
WO-2003035076-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO disclosed