SCHEMBL6650171

SCHEMBL6650171

O=CN1CCN(C(c2ccccc2)c2nc(C(=O)NCc3ccc(F)cc3)c(CO)c(=O)[nH]2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ATM Q13315 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
ERCC1 P07992 1/20 0.39
FEN1 P39748 1/20 0.39
ERCC4 Q92889 1/20 0.39
TP53 P04637 1/20 0.38
BRAF P15056 1/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR7 P34969 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CACNA2D1 P54289 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNB1 Q02641 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5127792 0.79 KMT2A (0.43) SMN1; SMN2MEN1KMT2AATMNPSR1
SCHEMBL6645450 0.79 SMN1; SMN2 (0.42) SMN1; SMN2MEN1KMT2AERCC1FEN1
SCHEMBL1150329 0.77 SMN1; SMN2 (0.47) SMN1; SMN2MEN1KMT2AATMNPSR1
SCHEMBL6647968 0.74 SMN1; SMN2 (0.46) SMN1; SMN2KMT2ANPSR1LMNAKDM4E
SCHEMBL6645878 0.72 ALDH1A1 (0.43) SMN1; SMN2MEN1KMT2AERCC1FEN1
SCHEMBL6651068 0.70 ERCC1 (0.52) SMN1; SMN2ERCC1FEN1ERCC4
SCHEMBL5118543 0.70 SMN1; SMN2 (0.44) SMN1; SMN2MEN1KMT2AATMNPSR1
SCHEMBL6646424 0.69 PARP1 (0.49) SMN1; SMN2MEN1KMT2A
SCHEMBL5118888 0.69 CALCA (0.45) SMN1; SMN2MEN1KMT2AATMNPSR1
SCHEMBL5118805 0.69 TP53 (0.46) SMN1; SMN2MEN1KMT2AATMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441735-A1 N-SUBSTITUTED HYDROXYPYRIMIDINONE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2004-08-04 EP disclosed
WO-2003035077-A1 N-SUBSTITUTED HYDROXYPYRIMIDINONE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO disclosed