SCHEMBL6651242

SCHEMBL6651242

FC(F)(F)Oc1ccc(-c2csc(-c3cnccc3C3CCCC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.42
ALOX5 P09917 1/20 0.40
EIF4E P06730 2/20 0.40
KDM4E B2RXH2 4/20 0.39
AR P10275 1/20 0.39
GABBR2 O75899 1/20 0.39
GABBR1 Q9UBS5 1/20 0.39
CYP19A1 P11511 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
MPL P40238 1/20 0.37
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
ADRB2 P07550 1/20 0.37
SCN5A Q14524 1/20 0.37
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 2/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
NPC1 O15118 1/20 0.36
HDAC3 O15379 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6627147 0.82 KDM4E (0.55) KDM4EARCYP19A1RAB9ANPC1
SCHEMBL6648183 0.81 CACNA1B (0.39) SCN9AEIF4EKDM4EARCYP19A1
SCHEMBL6654412 0.77 KDM4E (0.55) KDM4EARCYP19A1RAB9ASMN1; SMN2
SCHEMBL6627829 0.77 KDM4E (0.59) KDM4EARCYP19A1RAB9ASMN1; SMN2
SCHEMBL6649714 0.77 CYP19A1 (0.43) SCN9AALOX5EIF4EKDM4EAR
SCHEMBL6649359 0.77 CYP19A1 (0.46) SCN9AALOX5EIF4EKDM4EAR
SCHEMBL6649722 0.76 SREBF2 (0.46) SCN9AALOX5EIF4EKDM4EAR
SCHEMBL6649421 0.76 KDM4E (0.50) SCN9AKDM4EARCYP19A1RAB9A
SCHEMBL6651514 0.74 RAB9A (0.46) SCN9AKDM4EARCYP19A1RAB9A
SCHEMBL6649186 0.74 RAB9A (0.57) EIF4EKDM4ERAB9ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed