SCHEMBL6651312

SCHEMBL6651312

c1cc(C2CC2)c(-c2nc(-c3ccsc3)cs2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.42
AXL P30530 1/20 0.40
PBRM1 Q86U86 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
KDM4E B2RXH2 7/20 0.39
RAB9A P51151 5/20 0.39
NPC1 O15118 2/20 0.39
ALDH1A1 P00352 1/20 0.39
AR P10275 3/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 2/20 0.37
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6627829 0.82 KDM4E (0.59) CYP19A1KDM4ERAB9ANPC1ALDH1A1
SCHEMBL6654412 0.82 KDM4E (0.55) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6627147 0.80 KDM4E (0.55) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6651298 0.75 CYP19A1 (0.47) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6648609 0.75 CYP19A1 (0.44) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6648612 0.74 CYP19A1 (0.43) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6649421 0.74 KDM4E (0.50) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6651514 0.74 RAB9A (0.46) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6648183 0.74 CACNA1B (0.39) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL6653028 0.74 MAPT (0.50) RAB9ANPC1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed