SCHEMBL6651783

SCHEMBL6651783

O=C(c1cccs1)N1CCN(c2nccc(C(F)(F)F)n2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.70
SLC6A7 Q99884 3/20 0.63
PKM P14618 2/20 0.63
GAA P10253 3/20 0.52
KCNA5 P22460 1/20 0.52
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51
ADRB1 P08588 1/20 0.50
RBP4 P02753 1/20 0.50
SCD O00767 1/20 0.49
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
ALOX12 P18054 1/20 0.49
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RECQL P46063 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13149786 0.83 ALDH1A1 (1.00) ALDH1A1GAANPC1LMNAMAPT
SCHEMBL8356355 0.81 PKM (0.91) ALDH1A1SLC6A7PKMCA12CA1
SCHEMBL6650909 0.80 ALDH1A1 (0.70) ALDH1A1PKMGAAKCNA5NPC1
SCHEMBL5232026 0.79 SLC6A7 (0.68) ALDH1A1SLC6A7PKMCA12CA1
Hydrochloric Acid SCHEMBL6652741 0.79 ALDH1A1 (0.68) ALDH1A1PKMGAAKCNA5NPC1
SCHEMBL6650793 0.78 ALDH1A1 (0.71) ALDH1A1SLC6A7PKMGAACA12
Hypochlorous Acid SCHEMBL6652746 0.78 ALDH1A1 (0.67) ALDH1A1PKMGAAKCNA5NPC1
SCHEMBL6653095 0.78 ALDH1A1 (0.67) ALDH1A1GAANPC1LMNAMAPT
SCHEMBL6652874 0.77 PKM (0.72) ALDH1A1SLC6A7PKMCA12CA1
SCHEMBL3582132 0.77 SLC6A7 (1.00) ALDH1A1SLC6A7PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1202087-C Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments ESTEVE LABOR DR (ES) 2005-05-18 CN claimed
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP claimed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US claimed
CN-1268124-A Acyl-piperazinyl-pyrimidine derivatives, their preparation and use as medicaments ESTEVE LABOR DR (ES) 2000-09-27 CN claimed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP claimed