SCHEMBL6651834

SCHEMBL6651834

COc1cccc(C(=O)O)c1OCC=C(C)CCC=C(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.53
MAPT P10636 2/20 0.51
PTGES O14684 6/20 0.50
ALOX15 P16050 4/20 0.49
ICMT O60725 1/20 0.48
GMNN O75496 1/20 0.48
TRPA1 O75762 1/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48
CDK2 P24941 1/20 0.48
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
NDUFS8 O00217 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651830 1.00 MTNR1A (0.53) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL6652681 0.84 ICMT (0.56) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL31438947 0.84 ICMT (0.56) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL7033631 0.84 ICMT (0.56) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL31438944 0.84 ICMT (0.56) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL6653805 0.84 ICMT (0.56) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL4654953 0.83 ALOX15 (0.54) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL4654951 0.83 ALOX15 (0.54) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL15756532 0.83 ICMT (0.58) MTNR1AMAPTPTGESALOX15ICMT
SCHEMBL6652527 0.79 MAPT (0.63) MTNR1AMAPTPTGESALOX15NDUFS8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0875501-B1 Alkylenediamine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO CO LTD (JP) 2004-06-16 EP disclosed
EP-0802196-B1 Alkylenediamine derivatives as drugs for the treatment of ulcers and the inhibition of Helicobacter pylori SHISEIDO CO LTD (JP) 2001-08-29 EP disclosed
US-6043243-A Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO CO., LTD. (JP) 2000-03-28 US disclosed
US-6001880-A DISUBSTITUTED N-(2-DIALKYLAMINOETHYL)BENZAMIDE DERIVATIVES OF GIVEN FORMULA; ANTIBACTERIAL ACTIVITY AGAINST HELICOBACTER PYROLI, ADMINISTERING FOR THE PREVENTION OR CURE OF PEPTIC ULCERS SHISEIDO CO., LTD. (JP) 1999-12-14 US disclosed
US-5925667-A INHIBITS GROWTH OF HELICOBACTER PYLORI SHISEIDO CO., LTD. (JP) 1999-07-20 US disclosed
EP-0875501-A2 Alkylenediamine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1998-11-04 EP disclosed
EP-0869118-A1 Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1998-10-07 EP disclosed
US-5814634-A PEPTIC ULCERS, GASTRIC ULCERS SHISEIDO CO. LTD. (JP) 1998-09-29 US disclosed
EP-0802196-A1 Alkylenediamine derivative, antiulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1997-10-22 EP disclosed